From Data to Drugs: Strategies for Benefiting from the New Drug Discovery Technologies

This authoritative management report from New Drug Discovery and Scrip Reports will help you develop a viable technology strategy. Although investment in genomics alone runs into billions of dollars every year, this and other related drug discovery technologies have yet to bear fruit. Part of the problem lies in the flood of information which hampers senior executives in their strategy development.

Data to Drugs: Strategies for Benefiting from the New Drug Discovery Technologies explains the technologies, identifies short- and long-term commercial opportunities and assesses the companies at the cutting edge of drug discovery technology. It provides consultancy-level advice, guidance and analysis on every aspect of the technology-business interface.

It six in-depth sections the report equips you with a powerful set of insights into how best to manage technology and information. The analysis ranges from the technical challenges that remain to be solved using genomics and related technologies to their market impact, particularly the fruition of pharmacogenomics efforts.

Price: £995/$1,995/¥239,000
Ref: BS1015E
Pages: 160+
Published: July 1999

Table of Contents

List of Tables
List of Figures
About the Authors

Introduction
Facing the Future
What the New Technologies Offer
Overcoming Technological Limitations
Decision Points: Where Do We Go from Here?
Gaining a Strategic Edge

Chapter 1: The Continuing Revolution in Drug Discovery Technologies
Impact of New Drug Discovery Techniques
New Products
New Competitors
A New Suite of Complementary Platform Technologies
Genomics
Combinatorial Chemistry and High-Throughput
Screening
Bioinformatics
Functional Genomics
Proteomics
Pharmacogenomics
Changing Technical and Competitive Landscape
The Promise
The Challenge
Why the Need for New Technologies?
Economic Hurdles
The "Innovation Deficit"
Limitations of Traditional Drug Discovery
Technologies
Potential of New Technologies
Medical Breakthroughs
Market Potential
Current/Near-Term Products

Chapter 2: Gaining Access to New Technologies
Alternative Strategies for Bringing in New Technology
In-House Development
Discovery by In-House Scientists
Adaptation from Outside Sources
Partnerships with Academia
Partnerships with Smaller Technology Companies
Corporate Acquisitions
Organizing to Gain Access to New Technologies

Chapter 3: Technical Problems in Getting Results
Too Much Data, Not Enough Knowledge
Bridging the Gap between Data and Information
The Role of Bioinformatics
Uses of Bioinformatics
Requirements for Bioinformatics
Core Competencies
Critical Success Factors
Challenges
Getting from Sequences to Targets
The Lengthening Drug Discovery Pathway
Traditional and Evolving Technology
Structural Biology
Functional Genomics and Gene Chips
High-Throughput Screening
The Challenge of Genomics: So Many Targets, So Little Time

Chapter 4: Combinatorial Chemistry: Current Limitations, Future Promise
Current Issues
Use in High-Throughput Screening
Use in "Gene to Screen"
Need for Refinement
Types of Combinatorial Chemistry
Natural Products
Solid Phase Synthesis
Solution Phase Synthesis
Problems Associated with Combinatorial Chemistry
Purity and Structural Identification
Library Size and Differentiation
Hit-or-Miss Lead Generation
Solving the Diversity Dilemma
Computational Approaches
Redefining Diversity Space
New Approaches
Combinatorial Chemistry and the Genomics Challenge
Business Issues
New Directions

Chapter 5: Organizational and Strategic Challenges
Accessing and Assessing Outside Information
Information Sources
Sifting through the Deluge
Evaluating and Managing Partnerships
Partnership Objectives
Components for Integration: Build versus Buy
Dealing with Cultural and Size Differences
Partnerships with Biotech
Partnerships with Academia
Boosting R&D Innovation
The Cultural Challenge
The Impact of Mergers
Major Market Changes
Pharmacogenomics and Market Fragmentation
Curing Disease through Gene Therapy

Chapter 6: The New Frontier
Moving Toward Technological Solutions
Handling Raw Genomics Data
Academic Institutions
Industrial Sources
Identifying Disease-Causing Genes
Discovering New Drug Entities
SME Technology
LME Technology
Maximizing the Commercial Potential of the New Drug Discovery Technologies
Moving Past the Quick Fix
Positioning for Success
What the Future Holds

List of Tables

Table 1-1 Financial Clout of Leading Biotech Competitors

Table 1-2 Selected Leading Companies and Other Organizations Developing Drug Discovery Platform Technologies

Table 1-3 Breakdown of Drugs Approved by the FDA, 1995-1998

Table 1-4 Genomics-Based Therapeutics Currently in Clinical Trials

Table 2-1 Benefits and Drawbacks of Various Strategies for Acquiring New Technologies

Table 2-2 Organizations Involved in the SNP Consortium

Table 2-3 Selected Recent Deals Involving Genomics, Functional Genomics, or Pharmacogenomics

Table 2-4 Selected Recent Deals Involving Combinatorial Chemistry and/or High-Throughput Screening

Table 3-1 Fully Sequenced Microbial Genomes

Table 3-2 Exemplary Software Programs for Bioinformatics

Table 3-3 Companies Developing Gene Chip Technologies

Table 4-1 Characteristics of Different Types of Combinatorial Chemistry

Table 4-2 Requirements for Combinatorial Chemistry to Meet the Genomics Challenge

Table 5-1 Key Areas of Need for Timely Information

Table 5-2 Challenges in Gaining Timely Access to Critical Outside Information

Table 5-3 Sources of Information on Drug Discovery

Table 5-4 Goals of Partnerships with Biotech Companies and Academic Groups

Table 5-5 Key Factors in Make-or-Buy Decisions for Technology Platforms

Table 5-6 Big Pharma-Biotech Divisions That Can Affect the Success of Partnerships

Table 5-7 Pharmaceutical Satellite Laboratories in the Boston Area

Table 6-1 Interdisciplinary Life Science Centers Being Established by Academic Institutions

Table 6-2 Strategies for Bypassing the Limitations of Genomics and Molecular Diversity Technologies

Table 6-3 The Gap between Technology and Therapeutics: Small Molecule Drugs

Table 6-4 The Gap between Technology and Therapeutics: Protein Drugs

List of Figures

Figure 1-1 Transforming Effects of Biotechnology on the Pharmaceutical Industry of the 1980s

Figure 1-2 Role of Various Platform Technologies in the Genomics-Led Drug Discovery Process

Figure 1-3 Pre-Genomics Methods of Discovering New Leads

Figure 1-4 Pre-Genomics Sources of Potential New Drugs

Figure 1-5 Selected Patient Populations Targeted by Genomics-Based Therapies, 2005-2020

Figure 1-6 Market Potential of Genomics-Based Therapies for Selected Indications, 2005-2020

Figure 3-1 Investment Required for Different Stages in the Drug Discovery Pathway

Figure 3-2 Role of Bioinformatics in Linking Molecular Biology, Target Identification and Drug Discovery, and Computational Science

Figure 3-3 The Effect of Integrated Bioinformatics on Drug Discovery

Figure 3-4 The Traditional Drug Discovery Pathway

Figure 3-5 Reverse Integration in Drug Discovery

Figure 3-6 The Gene Chip Process

Figure 4-1 Current Pathway for Drug Discovery

Figure 4-2 Compressed Drug Discovery Process through Use of Chemical Ligands

Figure 4-3 Core and Building Block Assembly of Combinatorial Mixtures

Figure 4-4 Drug Diversity Space Based on Known Drugs

Figure 4-5 Proteomal Diversity Space: Beyond Current Drug Diversity Space

Figure 5-1 Moving from Information to Action MORPACE Pharma Group, Ltd.


© PJB Publications Ltd. 2000
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